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• Competitive antagonist
  ... [agonist]] for receptor [[binding site]]s on the same receptor. Sufficient antagonist will displace the agonist from the binding sites, resulting in a lower fre ... ... rcept and Y-intercept will each equal the [[dissociation constant]] of the antagonist.<ref name="prism"/>
  1 KB (140 words) - 18:40, 17 August 2008

Page text matches

• Competitive antagonist
  ... [agonist]] for receptor [[binding site]]s on the same receptor. Sufficient antagonist will displace the agonist from the binding sites, resulting in a lower fre ... ... rcept and Y-intercept will each equal the [[dissociation constant]] of the antagonist.<ref name="prism"/>
  1 KB (140 words) - 18:40, 17 August 2008
• Drug design
  ... tidine]], the prototypical [[H2-receptor antagonist|H₂-receptor antagonist]] from which the later members of the class were developed
  6 KB (827 words) - 06:06, 17 September 2008
• Cimetidine
  ... , /saɪ-}}) is a histamine [[H2-receptor antagonist|H₂-receptor antagonist]] that inhibits the production of acid in the [[stomach]]. It is largely ... ''Main article:[[H2-receptor antagonist]]''
  8 KB (1141 words) - 05:03, 25 August 2008
• Pharmacodynamics
  ... nding, receptors can elicit their normal action (agonist), blocked action (antagonist), or even action opposite to normal (inverse agonist).
  8 KB (1104 words) - 17:10, 29 August 2008
• Drug interaction
  ... namic]] properties of the drug, e.g. the co-administration of a [[receptor antagonist]] and an [[agonist]] for the same receptor.
  5 KB (686 words) - 10:34, 28 August 2008
• Biologics
  ... tis, ankylosing spondylitis, psoriatic arthritis monoclonal antibody TNF antagonist ... c arthritis, psoriasis recombinant human TNF-receptor fusion protein TNF antagonist
  10 KB (1491 words) - 09:52, 1 September 2008
• Chemicals with harmful effects
  ... dous" based on a rat LD50 of 80 mg/kg. It is a GABA-gated chloride channel antagonist, and a Ca2+, Mg2+ ATPase inhibitor. Both of these enzymes are involved in ...
  41 KB (6328 words) - 05:37, 2 September 2008
• Androgen
  ... ix 12 folds over the pocket to enclose the ligand PUBMED:12089231. When an antagonist is unbound, helix 12 is positioned away from the pocket in a way that inte ...
  7 KB (1027 words) - 07:00, 17 October 2008
• Steroid
  |ANTAGONIST |ANTAGONIST
  13 KB (1867 words) - 07:29, 18 October 2008
• Progestrone
  ... ptor (MR S810L) induces severe hypertension and switches progesterone from antagonist to agonist. Here we report the crystal structures of the ligand-binding do ... ... report multiple crystal structures of MR (NR3C2) bound to both agonist and antagonists. These structures combined with mutagenesis studies reveal that maximal r ...
  8 KB (1073 words) - 09:35, 19 February 2009
• Pregnenolone
  ... s a [[prohormone]]. Pregnenolone is a [[GABAB receptor|GABA_B]] antagonist and increases neurogenesis in the hippocampus.<ref name=Mayo2005>{{cite jo ...
  5 KB (687 words) - 09:34, 19 February 2009
• Aldosterone
  * [[Aldosterone antagonist]]
  17 KB (2332 words) - 11:48, 19 February 2009
• Serotonin
  [[5-HT3 antagonist|5-HT₃ antagonist]]s such as [[ondansetron]], [[granisetron]], and [[tropisetron]] are impor ... *Serotonin receptor agonists/antagonists
  38 KB (5178 words) - 12:28, 19 February 2009
• Dexamethasone
  ... the [[antiemetic]] effect of [[5-HT3 antagonist|5-HT₃ receptor antagonists]] like [[ondansetron]]. Dexamethasone is also used in certain [[hematolo ...
  13 KB (1840 words) - 10:44, 20 February 2009
• Genistein
  ... could be completely abolished by cotreatment of MCF-7 cells with estrogen antagonist ICI 182780 (1 microM) and tamoxifen (0.1 microM).
  11 KB (1547 words) - 09:12, 19 February 2009
• Lipoxin A4
  Lipoxins are high affinity [[receptor antagonist|antagonists]] to the cysteinyl leukotriene receptor type 1 (CysLT1) to which several ...
  8 KB (1055 words) - 06:32, 11 December 2009
• Cholecystokinin
  ... author = Shillabeer G, Davison JS | title = Proglumide, a cholecystokinin antagonist, increases gastric emptying in rats | journal = Am. J. Physiol. | volume = ...
  7 KB (948 words) - 06:42, 11 December 2009
• Follicle-stimulating hormone beta subunit
  ##[[GnRH antagonist]]
  6 KB (846 words) - 06:40, 17 February 2009
• Gonadoliberin-1
  ==Agonists and antagonists== ... late ([[GnRH agonist|GNRH1 agonist]]s) or suppress ([[GnRH antagonist|GNRH antagonist]]s) the gonadotropins. It is important to note that, through [[downregulat ...
  12 KB (1557 words) - 06:45, 11 December 2009
• Luteinizing hormone subunit beta (LSH-B) (LH-B)(Lutropin subunit beta)
  ##[[GnRH antagonist]]
  9 KB (1293 words) - 06:36, 17 February 2009

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