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• Diethylstilbestrol
  ... ostate cancer for over forty years, until the (much more expensive) [[GnRH agonist]] [[leuprolide]] was found to have efficacy similar to DES without estroge ... ... prostate cancer for over forty years, until the (much more expensive) GnRH agonist leuprolide was found to have efficacy similar to DES without estrogenic ef ...
  34 KB (4923 words) - 11:19, 20 February 2009
• Docking (molecular)
  ... the enzyme. If the protein is a receptor, ligand binding may result in [[agonist|agonism]] or [[Antagonism_(chemistry)|antagonism]]. Docking is most commo ...
  12 KB (1708 words) - 05:48, 17 September 2008
• Competitive antagonist
  ... ding site]]s on the same receptor. Sufficient antagonist will displace the agonist from the binding sites, resulting in a lower frequency of receptor activat ... ... pt and Y-intercept will each equal the [[dissociation constant]] of the antagonist.<ref name="prism"/>
  1 KB (140 words) - 18:40, 17 August 2008
• TGN1412
  ... ies|humanised monoclonal antibody]] that not only binds, but is a strong [[agonist]] for the [[CD28]] receptor of the [[immune system]]'s [[T cell]]s.<ref na ... | title = Superagonistic Anti-CD28 Antibody TGN1412 as a Potential Immunotherapeutic for the Trea ...
  29 KB (4350 words) - 08:44, 22 August 2008
• Clinical pharmacology
  ... r example, not just the biology of salbutamol, a beta2-adrenergic receptor agonist, but the peak flow meter|peak flow rate of both healthy volunteers and rea ...
  5 KB (777 words) - 07:18, 31 August 2008
• Pharmacodynamics
  ... ), blocked action (antagonist), or even action opposite to normal (inverse agonist). The graph shown represents the conc-response for two hypothetical receptor agonists, plotted in a semi-log fashion. The curve toward the left represents a hi ...
  8 KB (1104 words) - 17:10, 29 August 2008
• Drug interaction
  ... the drug, e.g. the co-administration of a [[receptor antagonist]] and an [[agonist]] for the same receptor.
  5 KB (686 words) - 10:34, 28 August 2008
• Androgen
  ... 12 folds over the pocket to enclose the ligand PUBMED:12089231. When an antagonist is unbound, helix 12 is positioned away from the pocket in a way that inte ... ... one and the estrogens estrone and estradiol. DHEA is also a potent sigma-1 agonist.
  7 KB (1027 words) - 07:00, 17 October 2008
• Steroid
  |AGONIST |AGONIST
  13 KB (1867 words) - 07:29, 18 October 2008
• Estradiol
  ... aromatase inhibitor]], or estrogen effects can be reduced with estrogen antagonists such as [[tamoxifen]]. Flaxseed is known to reduce estradiol.<ref>{{cite ... *Virtual and biomolecular screening converge on a selective agonist for GPR30
  21 KB (2912 words) - 05:26, 24 February 2009
• Liothyronine(T3)
  Cytosporone B is an agonist for nuclear orphan receptor Nur77
  11 KB (1699 words) - 10:11, 24 October 2008
• Progestrone
  ... omain of MR S810L in complex with progesterone and deoxycorticosterone, an agonist of both wild-type and mutant MRs.... ... ort multiple crystal structures of MR (NR3C2) bound to both agonist and antagonists. These structures combined with mutagenesis studies reveal that maximal r ...
  8 KB (1073 words) - 09:35, 19 February 2009
• Thaliporphine
  from plant Neolitsea konishii K; potent agonist of vascular smooth muscle contractions in the presence of calcium; RN give ...
  2 KB (259 words) - 06:05, 23 April 2009
• Dehydroepiandrosterone
  ... e]] and [[estradiol]]. DHEA is also a potent [[sigma-1 receptor|sigma-1]] agonist.<ref>Romieu, P., Martin-Fardon, R., Bowen, W. D., & Maurice, T. (2003). Si ...
  20 KB (2812 words) - 08:55, 20 February 2009
• Aldosterone
  ... la D, Almeida OF, Czéh B |title=The prototypic mineralocorticoid receptor agonist aldosterone influences neurogenesis in the dentate gyrus of the adrenalect ... * [[Aldosterone antagonist]]
  17 KB (2332 words) - 11:48, 19 February 2009
• Serotonin
  [[5-HT3 antagonist|5-HT₃ antagonist]]s such as [[ondansetron]], [[granisetron]], and [[tropisetron]] are impor ... ... id healing. Because of these effects, overdoses of serotonin, or serotonin agonist drugs, may cause acute or chronic pulmonary hypertension from pulmonary va ...
  38 KB (5178 words) - 12:28, 19 February 2009
• Epinephrine
  ... are mediated through adrenergic receptors. Epinephrine is a non-selective agonist of all adrenergic receptors. It activates α₁, α₂, ... ... c [[beta2-adrenergic receptor agonist|beta₂-adrenergic receptor agonist]]s are unavailable or ineffective.
  16 KB (2097 words) - 12:32, 19 February 2009
• 2-arachidonylglycerol
  ... Arachidonoylglycerol''' (2-AG), is an [[endocannabinoid]], an endogenous [[agonist]] of the [[CB1 receptor]].<ref name="pmid9285589">{{cite journal |author=S ... ... 'et al'' |title=2-Arachidonoylglycerol, an endogenous cannabinoid receptor agonist: identification as one of the major species of monoacylglycerols in variou ...
  7 KB (921 words) - 10:31, 10 December 2009
• Bisphenol A
  ... regulated kinase signaling in the rat cerebellar cortex: potent nongenomic agonist and endocrine disrupting activity of the xenoestrogen bisphenol A | journa ...
  48 KB (6845 words) - 04:51, 20 February 2009
• Follicle-stimulating hormone beta subunit
  ##[[GnRH antagonist]] ##[[GnRH agonist]] ([[downregulation]]).
  6 KB (846 words) - 06:40, 17 February 2009

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